| Title of Article |
Cross-coupling of Aromatic Aldehydes with N-(Amidobenzyl)benzotriazoles: An Alternative Route to α-Amidoketones |
| Date of Acceptance |
9 December 2017 |
| Journal |
| Title of Journal |
Letters in Organic Chemistry |
| Standard |
SCOPUS |
| Institute of Journal |
Bentham Science Publishers |
| ISBN/ISSN |
|
| Volume |
|
| Issue |
15 |
| Month |
April |
| Year of Publication |
2018 |
| Page |
838-844 |
| Abstract |
Several transition-metal-catalyzed reactions have been used to synthesize biologically active α-amidoketones. These approaches involve inconvenient conditions or expensive catalysts. Alternative attempts based on transition-metal-free catalysts have also been reported including cross-coupling reaction of aldehydes with acylimines in the presence of thiazolium salt as an organic catalyst. We report herein the use of N,N-dimethylbenzimidazolium iodide which is a safe and recyclable organic pre-catalyst, along with N-(amidobenzyl)benzotriazoles as activated N-acylimines for this cross-coupling reaction. |
| Keyword |
α-Amidoketones, N-(amidobenzyl)benzotriazoles, masked N-acylimines, N ,N-dimethylbenzimidazolium iodide, organic catalyst, aldehyde |
| Author |
|
| Reviewing Status |
มีผู้ประเมินอิสระ |
| Status |
ตีพิมพ์แล้ว |
| Level of Publication |
นานาชาติ |
| citation |
true |
| Part of thesis |
true |
| Attach file |
|
| Citation |
0
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Publication
Journal Publication
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